SCHEMBL18400347

SCHEMBL18400347

Fc1ccc(Cc2cnc(NC3(c4ccc5c(c4)OCO5)CC3)s2)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
CLPP Q16740 1/20 0.40
CFTR P13569 3/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
HPGD P15428 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ABL1 P00519 1/20 0.36
GPER1 Q99527 1/20 0.35
LMNA P02545 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
ULK1 O75385 1/20 0.35
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
MAP2K4 P45985 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18400325 0.92 HDAC3 (0.42) HDAC3HDAC1HDAC2HDAC6CFTR
SCHEMBL18400435 0.89 HDAC3 (0.42) HDAC3HDAC1HDAC2HDAC6CFTR
SCHEMBL18400383 0.85 HDAC3 (0.42) HDAC3HDAC1HDAC2HDAC6CFTR
SCHEMBL18400324 0.84 HDAC6 (0.41) HDAC3HDAC1HDAC2HDAC6CFTR
SCHEMBL12026803 0.83 CFTR (0.55) CFTR
SCHEMBL18400323 0.82 MEN1 (0.45) HDAC3HDAC1HDAC2HDAC6CFTR
SCHEMBL18400346 0.80 LMNA (0.48) HDAC3HDAC1HDAC2HDAC6CFTR
SCHEMBL18400321 0.80 MAPT (0.49) HDAC3HDAC1HDAC2HDAC6CFTR
SCHEMBL12026805 0.75 CFTR (0.55) CFTRLMNAMAPT
SCHEMBL2202153 0.75 ABL1 (0.46) CFTRKMT2AMEN1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9550761-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2017-01-24 US disclosed