SCHEMBL18409291

SCHEMBL18409291

CCc1cc(C#N)ncc1Nc1cc2c(ncn2C)c(N(Cc2ccc(OC)cc2OC)C(=O)C2CC2)n1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 10/20 0.37
JAK1 P23458 10/20 0.37
TYK2 P29597 10/20 0.37
JAK3 P52333 10/20 0.37
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
PIK3CA P42336 1/20 0.34
CHEK1 O14757 5/20 0.33
NR1H4 Q96RI1 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18409260 0.93 JAK2 (0.36) JAK2JAK1TYK2JAK3GABRG2
SCHEMBL18409113 0.88 ALDH1A1 (0.36) GABRG2GABRB3GABRA5PIK3CAMEN1
SCHEMBL18409289 0.86 JAK2 (0.41) JAK2JAK1TYK2JAK3NR1H4
SCHEMBL18409164 0.85 JAK2 (0.42) JAK2JAK1TYK2JAK3NR1H4
SCHEMBL18409541 0.84 PIK3CA (0.35) JAK2JAK1TYK2JAK3GABRG2
SCHEMBL18409180 0.84 TYK2 (0.35) JAK2JAK1TYK2JAK3GABRG2
SCHEMBL18409110 0.83 POLB (0.33) JAK2JAK1TYK2JAK3MEN1
SCHEMBL18409564 0.82 JAK2 (0.39) JAK2JAK1TYK2JAK3CHEK1
SCHEMBL18409360 0.82 MEN1 (0.36) GABRG2GABRB3GABRA5PIK3CAMEN1
SCHEMBL18409321 0.82 JAK2 (0.38) JAK2JAK1TYK2JAK3NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017012647-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS GALAPAGOS NV (BE) 2017-01-26 WO disclosed