SCHEMBL18436111

SCHEMBL18436111

COc1c(-c2ccc(N3C[C@@H](C)O[C@@H](C)C3)nc2)cnc2c(-c3ccc(C)cc3)cccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 2/20 0.45
PGR P06401 1/20 0.45
GPR183 P32249 1/20 0.45
ALDH1A1 P00352 3/20 0.41
GAA P10253 2/20 0.41
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ACVR1 Q04771 1/20 0.41
AOC3 Q16853 3/20 0.41
CNR2 P34972 2/20 0.40
TLR9 Q9NR96 1/20 0.40
TLR8 Q9NR97 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
KDM4E B2RXH2 2/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
EED O75530 1/20 0.38
SUZ12 Q15022 1/20 0.38
EZH2 Q15910 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21336856 1.00 SMO (0.45) SMOPGRGPR183ALDH1A1GAA
SCHEMBL18436839 1.00 SMO (0.45) SMOPGRGPR183ALDH1A1GAA
SCHEMBL18436802 0.93 ALDH1A1 (0.47) SMOPGRGPR183ALDH1A1GAA
SCHEMBL17127983 0.93 ALDH1A1 (0.47) SMOPGRGPR183ALDH1A1GAA
SCHEMBL18436713 0.93 ALDH1A1 (0.47) SMOPGRGPR183ALDH1A1GAA
SCHEMBL21336858 0.92 AOC3 (0.44) SMOPGRGPR183ALDH1A1GAA
SCHEMBL18436461 0.92 AOC3 (0.44) SMOPGRGPR183ALDH1A1GAA
SCHEMBL17127952 0.92 AOC3 (0.44) SMOPGRGPR183ALDH1A1GAA
SCHEMBL19001155 0.91 SMO (0.46) SMOPGRGPR183ALDH1A1ACVR1
SCHEMBL18436467 0.91 SMO (0.42) SMOPGRGPR183ALDH1A1ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-B1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO LTD (CN) 2019-09-11 EP disclosed
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed