SCHEMBL18436688

SCHEMBL18436688

CC(C)(O)c1ccc(N2CCNCC2(C)O)nc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMO Q99835 3/20 0.39
HRH3 Q9Y5N1 1/20 0.38
OGA O60502 1/20 0.37
OPRD1 P41143 1/20 0.35
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
HDAC11 Q96DB2 2/20 0.31
MAPT P10636 3/20 0.31
ALDH1A1 P00352 1/20 0.31
PANK3 Q9H999 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HSD11B1 P28845 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19001099 0.78 SMO (0.39) SMOHRH3OGACNR1CNR2
SCHEMBL19012353 0.78 SMO (0.39) SMOHRH3OGACNR1CNR2
SCHEMBL17128345 0.76 OGA (0.50) SMOHRH3OGAOPRD1MAPT
Hydrochloric Acid SCHEMBL28341448 0.75 OGA (0.49) SMOHRH3OGAOPRD1MAPT
SCHEMBL1471033 0.74 MAPT (0.41) CNR1CNR2HDAC11MAPTALDH1A1
SCHEMBL19012378 0.71 OGA (0.51) SMOHRH3OGAMAPTALDH1A1
SCHEMBL29977962 0.70 PIM1 (0.39) SMOHRH3OGAOPRD1MAPT
SCHEMBL18436110 0.70 PIM1 (0.39) SMOHRH3OGAOPRD1MAPT
SCHEMBL17128127 0.70 HTR2C (0.39) SMOHRH3OGAOPRD1
Hydrochloric Acid SCHEMBL29978429 0.69 PIM1 (0.39) SMOHRH3OGAOPRD1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-B1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO LTD (CN) 2019-09-11 EP disclosed
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed