SCHEMBL18436708

SCHEMBL18436708

CCc1c(-c2ccc(N3CC(C)O[C@H](C)C3)nc2)cnc2c(-c3ccc(C#N)cc3)cccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.40
SMO Q99835 2/20 0.39
PGR P06401 1/20 0.39
GPR183 P32249 1/20 0.39
LRRK2 Q5S007 2/20 0.39
HRH4 Q9H3N8 1/20 0.38
CNR2 P34972 1/20 0.38
MAP3K7 O43318 1/20 0.38
EED O75530 1/20 0.38
SUZ12 Q15022 1/20 0.38
EZH2 Q15910 1/20 0.38
ACVR1 Q04771 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
USP7 Q93009 2/20 0.36
TLR9 Q9NR96 1/20 0.36
TLR8 Q9NR97 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18436710 1.00 AOC3 (0.40) AOC3SMOPGRGPR183LRRK2
SCHEMBL18436183 1.00 AOC3 (0.40) AOC3SMOPGRGPR183LRRK2
SCHEMBL17127918 1.00 AOC3 (0.40) AOC3SMOPGRGPR183LRRK2
SCHEMBL18436282 0.90 HRH4 (0.40) LRRK2HRH4TDP1KDM4EALDH1A1
SCHEMBL21336668 0.90 HRH4 (0.40) LRRK2HRH4TDP1KDM4EALDH1A1
SCHEMBL17127857 0.90 HRH4 (0.40) LRRK2HRH4TDP1KDM4EALDH1A1
SCHEMBL17128422 0.88 CNR2 (0.46) AOC3SMOPGRGPR183LRRK2
SCHEMBL17127921 0.88 SMO (0.44) AOC3SMOPGRGPR183LRRK2
SCHEMBL18436199 0.88 SMO (0.44) AOC3SMOPGRGPR183LRRK2
SCHEMBL17128326 0.88 CNR2 (0.46) AOC3SMOPGRGPR183LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed