SCHEMBL21336668

SCHEMBL21336668

CCc1c(-c2ccc(N3CC(C)OC(C)C3)cc2)cnc2c(-c3ccc(C#N)cc3)cccc12

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.40
LRRK2 Q5S007 3/20 0.37
USP7 Q93009 2/20 0.36
PRKDC P78527 1/20 0.36
HRH3 Q9Y5N1 4/20 0.36
KDM1A O60341 3/20 0.35
TDP1 Q9NUW8 2/20 0.35
TSHR P16473 1/20 0.35
CYP11B2 P19099 1/20 0.35
MTOR P42345 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17127857 1.00 HRH4 (0.40) HRH4LRRK2USP7PRKDCHRH3
SCHEMBL18436282 1.00 HRH4 (0.40) HRH4LRRK2USP7PRKDCHRH3
SCHEMBL18436708 0.90 AOC3 (0.40) HRH4LRRK2USP7KDM1ATDP1
SCHEMBL18436710 0.90 AOC3 (0.40) HRH4LRRK2USP7KDM1ATDP1
SCHEMBL18436183 0.90 AOC3 (0.40) HRH4LRRK2USP7KDM1ATDP1
SCHEMBL17127918 0.90 AOC3 (0.40) HRH4LRRK2USP7KDM1ATDP1
SCHEMBL17127848 0.87 HRH4 (0.42) HRH4LRRK2PRKDCHRH3KDM1A
SCHEMBL21336664 0.87 HRH4 (0.42) HRH4LRRK2PRKDCHRH3KDM1A
SCHEMBL18436706 0.87 HRH4 (0.42) HRH4LRRK2PRKDCHRH3KDM1A
SCHEMBL17127887 0.87 HRH4 (0.42) HRH4LRRK2PRKDCHRH3KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-B1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO LTD (CN) 2019-09-11 EP disclosed