SCHEMBL18455270

SCHEMBL18455270

COc1cccc2cc(-c3n[nH]c(=O)[nH]3)nc(N)c12

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BTK Q06187 15/20 0.55
DCPS Q96C86 1/20 0.42
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
NPC1 O15118 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
TNKS O95271 1/20 0.37
PARP1 P09874 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18455263 0.81 BTK (0.49) BTKPARP1
Hydrochloric Acid SCHEMBL16008156 0.73 BTK (0.43) BTK
Hydrochloric Acid SCHEMBL16008154 0.73 BTK (0.43) BTK
SCHEMBL18455257 0.71 BTK (1.00) BTK
SCHEMBL1620226 0.67 ABCG2 (0.51) DCPSPDE3BPDE3AALDH1A1TNKS
SCHEMBL19497042 0.63 BTK (0.64) BTK
SCHEMBL18455658 0.63 BTK (0.74) BTK
SCHEMBL18455260 0.63 BTK (0.64) BTK
SCHEMBL30522124 0.63 GAA (0.56) DCPSALDH1A1GAA
SCHEMBL18526 0.63 GAA (0.56) DCPSALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3235814-A1 PYRIDINYL AND FUSED PYRIDINYL TRIAZOLONE DERIVATIVES Takeda Pharmaceutical Company Limited (JP) 2017-10-25 EP disclosed
EP-2970202-B1 PYRIDINYL AND FUSED PYRIDINYL TRIAZOLONE DERIVATIVES TAKEDA PHARMACEUTICALS CO (JP) 2017-02-01 EP disclosed