SCHEMBL1848089

SCHEMBL1848089

N#Cc1sc(NC(=O)C2CCCCC2)nc1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.48
BRAF P15056 5/20 0.48
KDR P35968 5/20 0.48
ADORA3 P0DMS8 2/20 0.46
RXFP1 Q9HBX9 3/20 0.46
ADORA2A P29274 4/20 0.45
ADORA1 P30542 3/20 0.45
CHEK1 O14757 1/20 0.43
IKBKB O14920 1/20 0.43
RAF1 P04049 1/20 0.43
PDGFA P04085 1/20 0.43
CDK1 P06493 1/20 0.43
PDGFRB P09619 1/20 0.43
CCNB1 P14635 1/20 0.43
CCNA2 P20248 1/20 0.43
FGFR3 P22607 1/20 0.43
CDK2 P24941 1/20 0.43
GSK3B P49841 1/20 0.43
MAP2K1 Q02750 1/20 0.43
TEK Q02763 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1846930 0.92 ADORA3 (0.53) JAK2BRAFKDRADORA3ADORA2A
SCHEMBL1854861 0.90 ADORA3 (0.48) JAK2BRAFKDRADORA3RXFP1
SCHEMBL3775335 0.90 ADORA3 (0.48) JAK2BRAFKDRADORA3RXFP1
SCHEMBL1854145 0.90 ADORA3 (0.48) JAK2BRAFKDRADORA3RXFP1
SCHEMBL3770544 0.88 KDR (0.47) JAK2BRAFKDRADORA3ADORA2A
SCHEMBL1848588 0.87 ADORA3 (0.58) ADORA3ADORA2AADORA1GSK3BKDM4E
SCHEMBL3764638 0.86 BRAF (0.42) JAK2BRAFKDRADORA3RXFP1
SCHEMBL1847530 0.86 ADORA3 (0.59) ADORA3ADORA2AADORA1GSK3BKDM4E
SCHEMBL1848517 0.85 KMT2A (0.48) JAK2ADORA3ADORA2AADORA1GSK3B
SCHEMBL1849615 0.85 MAPK14 (0.53) ADORA3ADORA2AADORA1MAPK14KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197860-B1 NEW COMPOUNDS AS ADENOSINE A1 RECEPTOR ANTAGONISTS PALOBIOFARMA SL (ES) 2011-05-25 EP claimed