SCHEMBL18488352

SCHEMBL18488352

CCC1CCCN(c2ccc(C(F)(F)F)cc2)C1CC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.39
CYP2C8 P10632 1/20 0.39
CYP2D6 P10635 1/20 0.39
CNR1 P21554 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
GAA P10253 2/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KDM2B Q8NHM5 1/20 0.38
BACE1 P56817 1/20 0.37
NOTUM Q6P988 1/20 0.36
DRD3 P35462 6/20 0.36
DRD2 P14416 4/20 0.36
KCNH2 Q12809 2/20 0.36
FPR1 P21462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9892989 0.81 FPR1 (0.44) CNR2CYP2C8CYP2D6CNR1CYP2C19
SCHEMBL28845226 0.80 AR (0.39) KMT2ADRD3DRD2
SCHEMBL16480461 0.75 AR (0.50) CNR2CYP2C8CYP2D6CNR1CYP2C19
SCHEMBL18490902 0.74 HRH3 (0.42) MAPTALDH1A1MAPK1NOTUM
SCHEMBL18490893 0.74 HRH3 (0.42) MAPTALDH1A1MAPK1NOTUM
SCHEMBL18488068 0.73 AKR1C3 (0.38) MAPTDRD3DRD2KCNH2
SCHEMBL9891844 0.73 CNR2 (0.45) CNR2CYP2C8CYP2D6CNR1CYP2C19
SCHEMBL21136651 0.72 BRD4 (0.50) CNR2CYP2C8CYP2D6CNR1CYP2C19
SCHEMBL18013246 0.72 BRD4 (0.50) CNR2CYP2C8CYP2D6CNR1CYP2C19
SCHEMBL20668703 0.71 FPR1 (0.58) CNR2FPR1FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3331886-B1 DOPAMINE D3 RECEPTOR ANTAGONISTS HAVING A BICYCLO MOIETY INDIVIOR UK LTD (GB) 2020-07-15 EP disclosed
WO-2017021920-A1 DOPAMINE D3 RECEPTOR ANTAGONISTS HAVING A BICYCLO MOIETY INDIVIOR UK LIMITED (GB) 2017-02-09 WO disclosed