SCHEMBL18489809

SCHEMBL18489809

CS(=O)(=O)NCc1cc(N)cc(F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.40
SCN9A Q15858 1/20 0.40
CYP19A1 P11511 2/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
TSHR P16473 1/20 0.35
RECQL P46063 1/20 0.35
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
CA1 P00915 1/20 0.34
CNR2 P34972 1/20 0.34
ALOX5 P09917 1/20 0.34
NSD2 O96028 2/20 0.33
CA12 O43570 1/20 0.33
CA7 P43166 1/20 0.33
CA14 Q9ULX7 1/20 0.33
PTGS2 P35354 1/20 0.33
GRIA2 P42262 1/20 0.33
CLK2 P49760 2/20 0.32
CLK3 P49761 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10312255 0.87 KMT2A (0.46) KMT2ASCN9ACYP19A1KDM4EPOLB
SCHEMBL17571471 0.81 KMT2A (0.41) KMT2ASCN9ACYP19A1KDM4EPOLB
SCHEMBL18474532 0.81 KMT2A (0.41) KMT2ASCN9ACYP19A1KDM4EPOLB
SCHEMBL15301413 0.79 KMT2A (0.40) KMT2ASCN9ACYP19A1KDM4EPOLB
SCHEMBL14785048 0.78 IDO1 (0.33) CA2CA1PTGS2
SCHEMBL18475990 0.78 KMT2A (0.39) KMT2ASCN9ACYP19A1KDM4EPOLB
SCHEMBL19022210 0.77 GRIA4 (0.39) KMT2AKDM4EPOLBTSHRRECQL
SCHEMBL17562440 0.77 KMT2A (0.38) KMT2ASCN9ACYP19A1KDM4EPOLB
SCHEMBL1542377 0.74 CYP19A1 (0.61) KMT2ACYP19A1KDM4EPOLBTSHR
SCHEMBL15218453 0.74 KMT2A (0.47) KMT2ACYP19A1KDM4EPOLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017023986-A1 3-(1H-INDOL-2-YL)-1H-INDAZOLES AND THERAPEUTIC USES THEREOF SAMUMED, LLC (US) 2017-02-09 WO disclosed