SCHEMBL1849337

SCHEMBL1849337

N#Cc1sc(NC(=O)C2CCCC2)nc1-c1ccccc1F

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.57
ADORA2A P29274 7/20 0.47
ADORA1 P30542 6/20 0.47
ALDH1A1 P00352 4/20 0.47
KDM4E B2RXH2 2/20 0.47
LMNA P02545 2/20 0.47
MAPT P10636 2/20 0.47
HPGD P15428 1/20 0.47
HTT P42858 1/20 0.47
NPC1 O15118 4/20 0.47
RAB9A P51151 4/20 0.47
ADORA2B P29275 3/20 0.47
POLB P06746 2/20 0.43
MEN1 O00255 1/20 0.43
PKM P14618 1/20 0.43
KMT2A Q03164 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
ABL1 P00519 3/20 0.42
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1847292 0.99 ADORA3 (0.56) ADORA3ADORA2AADORA1ALDH1A1KDM4E
SCHEMBL1848428 0.91 ADORA3 (0.65) ADORA3ADORA2AADORA1NPC1RAB9A
SCHEMBL1850969 0.91 ADORA3 (0.65) ADORA3ADORA2AADORA1NPC1RAB9A
SCHEMBL1846915 0.91 ADORA3 (0.65) ADORA3ADORA2AADORA1NPC1RAB9A
SCHEMBL1847852 0.90 ADORA3 (0.59) ADORA3ADORA2AADORA1ALDH1A1KDM4E
SCHEMBL1847849 0.90 ADORA3 (0.59) ADORA3ADORA2AADORA1ALDH1A1KDM4E
SCHEMBL1850635 0.90 ADORA3 (0.59) ADORA3ADORA2AADORA1ALDH1A1KDM4E
SCHEMBL1848849 0.90 ADORA3 (0.59) ADORA3ADORA2AADORA1ALDH1A1KDM4E
SCHEMBL1850636 0.90 ADORA3 (0.59) ADORA3ADORA2AADORA1ALDH1A1KDM4E
SCHEMBL1851737 0.87 ADORA3 (0.61) ADORA3ADORA2AADORA1ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197860-B1 NEW COMPOUNDS AS ADENOSINE A1 RECEPTOR ANTAGONISTS PALOBIOFARMA SL (ES) 2011-05-25 EP claimed