SCHEMBL1850315

SCHEMBL1850315

Clc1cc(Cl)cc(CN2CC=C(c3c[nH]c4ncccc34)CC2)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 1/20 0.63
SIGMAR1 Q99720 1/20 0.63
HTR1A P08908 13/20 0.56
SLC6A4 P31645 4/20 0.56
OPRM1 P35372 1/20 0.56
OPRK1 P41145 1/20 0.56
DRD2 P14416 11/20 0.55
HTR2A P28223 3/20 0.55
HTT P42858 1/20 0.55
ADRA1D P25100 1/20 0.54
ADRA1A P35348 1/20 0.54
ADRA1B P35368 1/20 0.54
DRD4 P21917 2/20 0.50
DRD3 P35462 2/20 0.50
CHEK1 O14757 2/20 0.47
MAP4K4 O95819 2/20 0.47
PIM1 P11309 2/20 0.47
PRKACA P17612 2/20 0.47
CLK2 P49760 2/20 0.47
GSK3B P49841 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1852412 0.88 TMEM97 (0.61) TMEM97SIGMAR1HTR1ASLC6A4OPRM1
SCHEMBL1849516 0.82 SIGMAR1 (0.73) TMEM97SIGMAR1HTR1ASLC6A4OPRM1
SCHEMBL13502652 0.81 SIGMAR1 (0.68) TMEM97SIGMAR1HTR1ASLC6A4DRD2
SCHEMBL1855275 0.81 CHEK1 (0.63) TMEM97SIGMAR1HTR1ASLC6A4ADRA1D
SCHEMBL31279383 0.77 TMEM97 (0.51) TMEM97SIGMAR1HTR1ASLC6A4OPRM1
SCHEMBL13064304 0.75 TMEM97 (0.59) TMEM97SIGMAR1HTR1ASLC6A4DRD2
SCHEMBL2064431 0.75 SLC6A4 (0.64) TMEM97SIGMAR1HTR1ASLC6A4ADRA1D
SCHEMBL31279305 0.74 TMEM97 (0.49) TMEM97SIGMAR1HTR1ASLC6A4OPRM1
SCHEMBL1853604 0.73 SIGMAR1 (0.69) TMEM97SIGMAR1HTR1ASLC6A4DRD2
SCHEMBL31338246 0.73 TMEM97 (0.51) TMEM97SIGMAR1HTR1ASLC6A4OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323659-A1 COMPOUNDS USEFUL AS INHIBITORS OF PROTEIN KINASES Abbott Laboratories (US) 2011-05-25 EP disclosed
WO-2010017150-A1 COMPOUNDS USEFUL AS INHIBITORS OF PROTEIN KINASES ABBOTT LABORATORIES (US) 2010-02-11 WO disclosed