SCHEMBL18508243

SCHEMBL18508243

Nc1cc(Br)ccc1NC(=O)C1CCC(F)(F)CC1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 4/20 0.59
HDAC1 Q13547 6/20 0.48
HDAC2 Q92769 6/20 0.48
HDAC3 O15379 5/20 0.48
KMT2A Q03164 2/20 0.44
POLB P06746 1/20 0.44
ALDH1A1 P00352 1/20 0.43
ABL1 P00519 1/20 0.43
TSHR P16473 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15746313 0.85 AAK1 (0.74) AAK1HDAC1HDAC2HDAC3KMT2A
SCHEMBL24969552 0.80 KMT2A (0.55) HDAC1HDAC2HDAC3KMT2APOLB
SCHEMBL30152391 0.80 KMT2A (0.55) HDAC1HDAC2HDAC3KMT2APOLB
SCHEMBL15111081 0.78 AAK1 (0.61) AAK1HDAC1HDAC2HDAC3KMT2A
SCHEMBL20096319 0.76 KDM4E (0.41) AAK1HDAC1HDAC2MAPT
SCHEMBL7604703 0.76 HDAC1 (0.63) AAK1HDAC1HDAC2HDAC3
SCHEMBL15594368 0.76 KMT2A (0.68) AAK1KMT2APOLBALDH1A1ABL1
SCHEMBL18496269 0.75 ABL1 (0.41) AAK1ABL1
SCHEMBL18496263 0.75 ABL1 (0.39) AAK1KMT2APOLBALDH1A1ABL1
SCHEMBL18496295 0.75 ABL1 (0.41) AAK1ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3334719-B1 SUBSTITUTED BENZIMIDAZOLES, THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS NEOMED INST (CA) 2021-09-15 EP disclosed
WO-2017024412-A1 SUBSTITUTED BENZIMIDAZOLES, THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS NEOMED INSTITUTE (CA) 2017-02-16 WO disclosed