SCHEMBL18516652

SCHEMBL18516652

COc1ccccc1NC(=O)CC(=O)Nc1ccc(Oc2ccnc3cc(-c4cccc(CC5CCCCOCCC5)c4)sc23)c(F)c1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.61
KDR P35968 19/20 0.61
AURKA O14965 1/20 0.45
FPR1 P21462 1/20 0.45
FPR3 P25089 1/20 0.45
GPR183 P32249 1/20 0.45
SMO Q99835 1/20 0.45
GPR35 Q9HC97 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL895974 0.86 KDR (0.65) METKDR
SCHEMBL308497 0.84 MET (0.69) METKDR
SCHEMBL306602 0.80 MET (0.67) METKDR
SCHEMBL306770 0.80 MET (0.69) METKDR
SCHEMBL18516387 0.80 MET (0.72) METKDR
SCHEMBL895849 0.80 KDR (0.63) METKDR
SCHEMBL896686 0.80 MET (0.64) METKDR
SCHEMBL306489 0.79 MET (0.68) METKDR
SCHEMBL307199 0.79 MET (0.68) METKDR
SCHEMBL307499 0.78 MET (0.69) METKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957498-B1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING METHYLGENE INC (CA) 2017-02-15 EP disclosed