SCHEMBL1851748

SCHEMBL1851748

CCOC(=O)c1cccc(-c2ccc(Cl)c3cc(CBr)sc23)c1.CCOC(=O)c1cccc(-c2ccc(Cl)c3cc(Cc4ccc(F)c(F)c4)sc23)c1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 5/20 0.44
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
CYP1A2 P05177 1/20 0.35
PRKDC P78527 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3217605 0.96 GPR52 (0.47) GPR52TP53POLBHPGDRAB9A
SCHEMBL1864780 0.93 GPR52 (0.50) GPR52CYP4F2CYP4A11TP53POLB
SCHEMBL1851227 0.92 GPR52 (0.44) GPR52TP53POLBHPGDRAB9A
SCHEMBL3206666 0.89 GPR52 (0.54) GPR52CYP4F2CYP4A11TP53POLB
SCHEMBL1854682 0.89 TP53 (0.43) CYP4F2CYP4A11TP53POLBHPGD
SCHEMBL1850740 0.87 GPR52 (0.49) GPR52TP53POLBHPGDRAB9A
SCHEMBL1854655 0.85 GPR52 (0.51) GPR52CYP4F2CYP4A11TP53POLB
SCHEMBL1854211 0.85 TP53 (0.41) CYP4F2CYP4A11TP53POLBHPGD
SCHEMBL1852550 0.85 GPR52 (0.46) GPR52CYP4F2CYP4A11TP53POLB
SCHEMBL1851960 0.84 GPR52 (0.55) GPR52TP53POLBHPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed