SCHEMBL18520113

SCHEMBL18520113

CCc1cnn2c(=O)[nH]cnc12

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 13/20 0.41
PDE4A P27815 13/20 0.41
PDE4B Q07343 13/20 0.41
PDE4C Q08493 13/20 0.41
PDE4D Q08499 13/20 0.41
ALDH1A1 P00352 1/20 0.40
ADORA2B P29275 7/20 0.39
ADORA3 P0DMS8 1/20 0.39
HPGD P15428 1/20 0.39
ADORA1 P30542 1/20 0.39
BLM P54132 1/20 0.39
PDE3A Q14432 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CHEK1 O14757 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
ATAD2 Q6PL18 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21539441 0.85 ALDH1A1 (0.36) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL18520818 0.79 ALDH1A1 (0.42) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL4165610 0.79 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL18520991 0.77 ALDH1A1 (0.40) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL21137393 0.76 ADORA2A (0.36) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL4163748 0.76 PNP (0.32) ALDH1A1
SCHEMBL4165764 0.76 PNP (0.34) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL4168419 0.75 ALDH1A1 (0.34) ALDH1A1BLM
SCHEMBL21273229 0.75 ALDH1A1 (0.39) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL867287 0.75 KDR (0.42) ADORA2APDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017027646-A1 CYCLIC DI-NUCLEOTIDE COMPOUNDS AS STING AGONISTS MERCK SHARP & DOHME CORP. (US) 2017-02-16 WO disclosed