SCHEMBL1852548

SCHEMBL1852548

O=C(NCCO)c1cccc(-c2cccc3nn(Cc4ccc(F)cc4)cc23)c1.O=C(O)c1cccc(-c2cccc3nn(Cc4ccc(F)cc4)cc23)c1

nearest known ligand 0.70

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 6/20 0.70
PTGER4 P35408 6/20 0.47
FYN P06241 4/20 0.41
ADORA3 P0DMS8 1/20 0.40
ADORA2B P29275 1/20 0.40
HDAC6 Q9UBN7 1/20 0.39
PPARG P37231 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3217594 0.96 GPR52 (0.75) GPR52PTGER4FYNADORA3ADORA2B
SCHEMBL1851055 0.91 GPR52 (0.65) GPR52PTGER4FYNADORA3ADORA2B
SCHEMBL3206799 0.90 GPR52 (0.78) GPR52FYNADORA3ADORA2BHDAC6
SCHEMBL1850248 0.90 GPR52 (0.54) GPR52PTGER4ADORA3ADORA2BHDAC6
SCHEMBL1853937 0.89 GPR52 (0.72) GPR52PTGER4FYNADORA3ADORA2B
SCHEMBL1849152 0.88 GPR52 (0.79) GPR52PTGER4FYN
SCHEMBL3207391 0.88 GPR52 (0.75) GPR52PTGER4FYN
SCHEMBL1850562 0.87 GPR52 (0.72) GPR52PTGER4FYNADORA3ADORA2B
SCHEMBL3209129 0.87 GPR52 (0.69) GPR52FYNADORA3ADORA2B
SCHEMBL1849610 0.86 GPR52 (0.93) GPR52PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed