SCHEMBL18525487

SCHEMBL18525487

C#Cc1cc(C)nc(C2CCC2)c1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.34
CTSS P25774 2/20 0.34
HRH4 Q9H3N8 5/20 0.33
CHRNA1 P02708 3/20 0.31
CHRNB4 P30926 3/20 0.31
CHRNA3 P32297 3/20 0.31
CHRNB2 P17787 2/20 0.31
CHRNA4 P43681 2/20 0.31
CHRNG P07510 1/20 0.31
CHRNB1 P11230 1/20 0.31
CHRND Q07001 1/20 0.31
CHRNA2 Q15822 1/20 0.31
DRD2 P14416 1/20 0.31
DRD1 P21728 1/20 0.31
DRD4 P21917 1/20 0.31
DRD5 P21918 1/20 0.31
DRD3 P35462 1/20 0.31
TLR8 Q9NR97 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18489390 0.83 CTSK (0.43) CTSKCTSSHRH4DRD2DRD3
SCHEMBL18489380 0.79 CTSK (0.47) CTSKCTSSHRH4
SCHEMBL18489386 0.75 CTSK (0.39) CTSKCTSS
SCHEMBL3720436 0.74 CYP1A1 (0.39)
SCHEMBL12250775 0.72 HRH4 (0.42) CTSKCTSSHRH4TLR8
SCHEMBL19531941 0.69 HRH4 (0.40) CTSKCTSSHRH4TLR8
Hydrochloric Acid SCHEMBL28371163 0.69 HRH4 (0.36) CTSKCTSSHRH4
SCHEMBL18497852 0.69 RAMP1 (0.38) CTSKCTSSHRH4TLR8
SCHEMBL25406682 0.68 TLR8 (0.41) TLR8
Hydrochloric Acid SCHEMBL18489419 0.68 RAMP1 (0.37) CTSKCTSSHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017027343-A1 CGRP RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2017-02-16 WO disclosed