SCHEMBL18526772

SCHEMBL18526772

COC(=O)NC(CC(=O)O)Cc1ccccc1F

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.45
CTSK P43235 1/20 0.45
MME P08473 2/20 0.44
KMT2A Q03164 1/20 0.44
CTSA P10619 1/20 0.42
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
PIN1 Q13526 1/20 0.40
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40
MMEL1 Q495T6 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
ALDH1A1 P00352 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
CXCL8 P10145 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL755370 1.00 CTSS (0.45) CTSSCTSKMMEKMT2ACTSA
SCHEMBL890178 0.89 CTSS (0.42) CTSSCTSKKMT2APPARGPPARA
SCHEMBL888773 0.88 CTSS (0.41) CTSSCTSKKMT2APPARGPPARA
SCHEMBL30753714 0.87 CTSS (0.60) CTSSCTSK
SCHEMBL4896150 0.87 CTSS (0.60) CTSSCTSK
SCHEMBL3997764 0.87 CTSS (0.60) CTSSCTSK
SCHEMBL17015 0.87 CTSS (0.60) CTSSCTSK
SCHEMBL8917906 0.86 CTSS (0.41) CTSSCTSKKMT2APPARGPPARA
SCHEMBL8290320 0.86 CTSS (0.41) CTSSCTSKMMEKMT2ACTSA
SCHEMBL14034476 0.85 MME (0.48) CTSSCTSKMMEKMT2ACTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2601188-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-10-18 EP disclosed
EP-2513091-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-04-12 EP disclosed
EP-2499132-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-02-15 EP disclosed