SCHEMBL18529253

SCHEMBL18529253

O=C(NC(=O)c1ccccc1)Nc1ncc([N+](=O)[O-])s1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 8/20 0.70
KMT2A Q03164 8/20 0.70
NPC1 O15118 7/20 0.70
RAB9A P51151 7/20 0.70
MAPT P10636 4/20 0.70
HTT P42858 3/20 0.70
ALDH1A1 P00352 2/20 0.70
LMNA P02545 2/20 0.70
SMN1; SMN2 Q16637 2/20 0.70
ATG4B Q9Y4P1 7/20 0.65
CDK2 P24941 1/20 0.65
GSK3A P49840 1/20 0.65
GSK3B P49841 1/20 0.65
DYRK1A Q13627 1/20 0.65
HIPK4 Q8NE63 1/20 0.65
CLK4 Q9HAZ1 1/20 0.65
STAT3 P40763 5/20 0.62
PKM P14618 3/20 0.62
NPSR1 Q6W5P4 2/20 0.61
THRB P10828 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1804666 0.89 NPC1 (0.76) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL18529265 0.88 NPC1 (0.60) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL376089 0.83 MEN1 (1.00) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL30142801 0.81 STAT3 (0.69) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL27135410 0.81 STAT3 (0.69) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL1394887 0.79 ATG4B (1.00) ATG4BCDK2GSK3AGSK3BDYRK1A
SCHEMBL29056922 0.78 STAT3 (0.77) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL16687501 0.78 NPC1 (0.77) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL12974167 0.77 NPC1 (0.78) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL30142722 0.77 STAT3 (0.75) MEN1KMT2ANPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017027984-A1 COMPOUNDS AND METHODS FOR TREATMENT OF CANCER BY INHIBITING ATG4B AND BLOCKING AUTOPHAGY SIMON FRASER UNIVERSITY (CA) 2017-02-23 WO disclosed
WO-2017027984-A1 COMPOUNDS AND METHODS FOR TREATMENT OF CANCER BY INHIBITING ATG4B AND BLOCKING AUTOPHAGY SIMON FRASER UNIVERSITY (CA) 2017-02-23 WO disclosed