SCHEMBL1852989

SCHEMBL1852989

CCOC(=O)Oc1ccc(C(=O)Nc2cc(CCc3cccc(OC)c3)n[nH]2)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.42
ROCK1 Q13464 4/20 0.41
ROCK2 O75116 3/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
TP53 P04637 2/20 0.40
NR3C2 P08235 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
MAPT P10636 1/20 0.38
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
CXCR1 P25024 1/20 0.37
CXCR2 P25025 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
PRKACA P17612 1/20 0.37
GRK5 P34947 1/20 0.37
PRKX P51817 1/20 0.37
PRKCQ Q04759 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1859162 0.93 ABCB1 (0.44) ABCB1ROCK1ROCK2RAB9ANR3C2
SCHEMBL1856714 0.90 ABCB1 (0.44) ABCB1ROCK1ROCK2RAB9ANR3C2
SCHEMBL62554 0.90 ABCB1 (0.47) ABCB1ROCK1ROCK2RAB9ANR3C2
SCHEMBL63192 0.86 ABCB1 (0.43) ABCB1ROCK1ROCK2NPC1RAB9A
SCHEMBL64112 0.86 ABCB1 (0.44) ABCB1ROCK1ROCK2RAB9ANR3C2
SCHEMBL65150 0.86 ABCB1 (0.49) ABCB1ROCK1ROCK2NPC1RAB9A
SCHEMBL1853874 0.85 ABCB1 (0.45) ABCB1ROCK1ROCK2NPC1RAB9A
SCHEMBL65051 0.84 HDAC1 (0.44) ABCB1ROCK1ROCK2NPC1RAB9A
SCHEMBL62361 0.84 ABCB1 (0.47) ABCB1ROCK1ROCK2RAB9ANR3C2
SCHEMBL64118 0.84 KCNQ3 (0.52) ABCB1ROCK1ROCK2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125748-B1 ACYLAMINOPYRAZOLES AS FGFR INHIBITORS ASTRAZENECA AB (SE) 2011-05-25 EP claimed