SCHEMBL18530871

SCHEMBL18530871

CC(C)C(=O)C1CCc2cc(-n3cnnn3)ccc21

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 16/20 0.50
ALDH1A1 P00352 2/20 0.46
HPGD P15428 1/20 0.46
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2731505 0.85 KCNJ1 (0.53) KCNJ1
SCHEMBL17268268 0.84 PPARD (0.43) KCNJ1
SCHEMBL15832633 0.79 KCNJ1 (0.47) KCNJ1ALDH1A1HPGD
SCHEMBL4549512 0.78 KCNJ1 (0.58) KCNJ1
SCHEMBL15825922 0.77 TP53 (0.49) KCNJ1TP53
Hydrochloric Acid SCHEMBL15192604 0.77 KCNJ1 (0.57) KCNJ1
SCHEMBL15825095 0.73 NOTUM (0.43) KCNJ1ALDH1A1HPGD
SCHEMBL19597281 0.71 KCNJ1 (0.72) KCNJ1
SCHEMBL19002833 0.70 MTNR1A (0.47)
Lithium Ion SCHEMBL15878970 0.68 KCNJ1 (0.40) KCNJ1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9573961-B2 Inhibitors of the renal outer medullary potassium channel MERCK SHARP & DOHME CORP. (US) 2017-02-21 US disclosed