SCHEMBL185329

SCHEMBL185329

[CH2]c1ncc(Nc2ccc(Cl)cc2C(F)(F)F)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
KDM4E B2RXH2 2/20 0.37
KCNQ3 O43525 2/20 0.37
KCNQ2 O43526 2/20 0.37
KCNE1 P15382 2/20 0.37
KCNQ1 P51787 2/20 0.37
IDO1 P14902 1/20 0.36
TGFBR1 P36897 1/20 0.36
STK17A Q9UEE5 2/20 0.35
STK17B O94768 1/20 0.35
NPC1 O15118 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL672412 0.81 DHODH (0.44) DHODHULK1DHFRSYKEGFR
SCHEMBL185709 0.81 STK17A (0.38) RAB9ACYP1A2CYP2D6CYP2C19SMN1; SMN2
Hydrochloric Acid SCHEMBL15456151 0.80 STK17A (0.37) RAB9ACYP1A2CYP2D6CYP2C19SMN1; SMN2
Hydrochloric Acid SCHEMBL2806736 0.80 STK17A (0.37) RAB9ACYP1A2CYP2D6CYP2C19SMN1; SMN2
SCHEMBL185783 0.79 RAB9A (0.38) RAB9ACYP1A2CYP2D6CYP2C19SMN1; SMN2
SCHEMBL2806482 0.76 RAB9A (0.44) RAB9ACYP1A2CYP2D6CYP2C19SMN1; SMN2
SCHEMBL185820 0.74 RAB9A (0.39) RAB9ACYP1A2CYP2D6CYP2C19SMN1; SMN2
SCHEMBL186155 0.73 CHEK1 (0.47)
SCHEMBL28794901 0.73 RAB9A (0.39) RAB9ACYP1A2CYP2D6CYP2C19SMN1; SMN2
SCHEMBL185410 0.73 RAB9A (0.39) RAB9ACYP1A2CYP2D6CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed