SCHEMBL18534006

SCHEMBL18534006

COC(CCCc1cc(NCc2ccc(Cl)cc2Cl)nc(N2CCNCC2)n1)OC

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 15/20 0.45
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
DPP4 P27487 1/20 0.39
INPPL1 O15357 1/20 0.38
HTR2A P28223 1/20 0.37
HTR7 P34969 1/20 0.37
HTR6 P50406 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16692263 0.81 CCR4 (0.45) CCR4ESR1ESR2DPP4INPPL1
SCHEMBL16258707 0.79 CCR4 (0.55) CCR4ESR1ESR2DPP4INPPL1
SCHEMBL16692262 0.75 CCR4 (0.46) CCR4ESR1ESR2MEN1KMT2A
SCHEMBL16242164 0.72 CCR4 (0.45) CCR4
SCHEMBL16242132 0.69 CCR4 (0.44) CCR4MEN1KMT2A
SCHEMBL16242226 0.67 CCR4 (0.45) CCR4
SCHEMBL13780220 0.67 HRH4 (0.43) CCR4ESR1ESR2KMT2AHTR2A
SCHEMBL16242162 0.67 CCR4 (0.44) CCR4
SCHEMBL16242163 0.67 CCR4 (0.41) CCR4MEN1KMT2A
SCHEMBL16258760 0.66 CCR4 (0.44) CCR4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2805947-B1 PIPERAZINYL PYRIMIDINE DERIVATIVES, PREPARATION METHOD AND USE THEREOF INST PHARMACOLOGY & TOXICOLOGY ACAD MILITARY MEDICAL SCIENCES PLA CHINA (CN) 2017-02-22 EP disclosed