SCHEMBL18534945

SCHEMBL18534945

C[C@@H](N[S+]([O-])C(C)(C)C)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.48
NOS3 P29474 1/20 0.38
NOS2 P35228 1/20 0.38
KCNN4 O15554 1/20 0.35
NPSR1 Q6W5P4 2/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
AR P10275 1/20 0.34
TRPV3 Q8NET8 1/20 0.33
IDH2 P48735 1/20 0.33
ALDH1A1 P00352 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
GAA P10253 1/20 0.32
MAPK1 P28482 1/20 0.32
ADRB1 P08588 1/20 0.31
ACACB O00763 1/20 0.31
DLK1 P80370 1/20 0.31
MAP3K12 Q12852 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14751140 1.00 ADRB2 (0.48) ADRB2NOS3NOS2KCNN4NPSR1
SCHEMBL25368832 0.87 ADRB2 (0.39) ADRB2
SCHEMBL25368834 0.87 ADRB2 (0.39) ADRB2
SCHEMBL25368946 0.87 ADRB2 (0.39) ADRB2
SCHEMBL29598075 0.87 ADRB2 (0.39) ADRB2
SCHEMBL2714728 0.82 CYP2C9 (0.38) ADRB2MAPTALDH1A1
SCHEMBL2714730 0.82 CYP2C9 (0.38) ADRB2MAPTALDH1A1
SCHEMBL2713443 0.82 CYP2C9 (0.38) ADRB2MAPTALDH1A1
SCHEMBL28392932 0.82 CYP2C9 (0.38) ADRB2MAPTALDH1A1
SCHEMBL24529689 0.80 KDM4C (0.34) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2763990-B1 PYRROLOPYRAZINE KINASE INHIBITORS HOFFMANN LA ROCHE (CH) 2017-02-22 EP disclosed