SCHEMBL18540693

SCHEMBL18540693

CC(C)(C)[Si](C)(C)Oc1cccc(C(=O)c2cc(Br)cc(Br)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 6/20 0.40
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA9 Q16790 2/20 0.39
MAOB P27338 2/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
MAOA P21397 1/20 0.37
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
ALOX15 P16050 1/20 0.37
HTT P42858 1/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18529823 0.93 MAOB (0.43) STSHSP90AA1HSP90AB1CA12CA1
SCHEMBL30785086 0.87 STS (0.50) STSHSP90AA1HSP90AB1ALDH1A1CYP1A2
SCHEMBL18529878 0.85 CA12 (0.38) HSP90AA1HSP90AB1CA12CA1CA9
SCHEMBL18540604 0.83 CA12 (0.36) HSP90AA1HSP90AB1CA12CA1CA9
SCHEMBL2989104 0.81 AKR1C3 (0.53) HSP90AA1HSP90AB1CA12CA1CA9
SCHEMBL341880 0.81 KMT2A (0.53) HSP90AA1HSP90AB1CA12CA1CA9
SCHEMBL5188852 0.81 MAPT (0.55) HSP90AA1HSP90AB1CA12CA1CA9
SCHEMBL2676116 0.80 HSP90AA1 (0.41) HSP90AA1HSP90AB1CA12CA1CA9
SCHEMBL5155346 0.80 AKR1C2 (0.44) ALDH1A1
SCHEMBL5156418 0.80 AKR1C2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017030983-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF CATHEPSINS MATEON THERAPEUTICS, INC. (US) 2017-02-23 WO disclosed