SCHEMBL18540604

SCHEMBL18540604

CC(C)(C)[Si](C)(C)Oc1cccc(C(=N)c2cc(Br)cc(Br)c2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.36
CA1 P00915 4/20 0.36
CA9 Q16790 4/20 0.36
PRSS1 P07477 3/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
C1S P09871 1/20 0.35
F2 P00734 2/20 0.33
F10 P00742 2/20 0.33
MAOB P27338 2/20 0.32
MAOA P21397 1/20 0.32
TP53 P04637 1/20 0.32
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
NPC1 O15118 1/20 0.31
POLB P06746 1/20 0.31
CYP2C9 P11712 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18540693 0.83 STS (0.40) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL18529823 0.79 MAOB (0.43) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL232409 0.75 CA12 (0.45) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL2989104 0.75 AKR1C3 (0.53) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL16554270 0.75 CA12 (0.40) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL341880 0.75 KMT2A (0.53) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL7706827 0.75 CA1 (0.50) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL2676116 0.74 HSP90AA1 (0.41) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL4576483 0.74 CA12 (0.44) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL2981524 0.74 HSP90AA1 (0.43) CA12CA1CA9HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017030983-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF CATHEPSINS MATEON THERAPEUTICS, INC. (US) 2017-02-23 WO disclosed