SCHEMBL18543778

SCHEMBL18543778

NCCc1ncc(I)cn1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 5/20 0.35
HRH1 P35367 4/20 0.35
TAAR1 Q96RJ0 1/20 0.33
HRH3 Q9Y5N1 4/20 0.32
HRH2 P25021 3/20 0.32
TSHR P16473 2/20 0.32
LMNA P02545 1/20 0.32
MIF P14174 1/20 0.32
APEX1 P27695 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CHRNA7 P36544 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.31
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
MTOR P42345 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4606399 0.75 APLNR (0.50) HRH4HRH1TAAR1HRH3HRH2
SCHEMBL2002429 0.75 TAAR1 (0.41) HRH4HRH1TAAR1HRH3HRH2
SCHEMBL9999635 0.75 HRH4 (0.45) HRH4HRH1TAAR1HRH3HRH2
Hydrochloric Acid SCHEMBL1396035 0.73 APLNR (0.48) HRH4HRH1TAAR1HRH3HRH2
SCHEMBL15332698 0.71 HRH1 (0.33) HRH4HRH1HRH3HRH2TSHR
SCHEMBL1086870 0.70
Hydrochloric Acid SCHEMBL29956780 0.70 HRH4 (0.32) HRH4HRH1HRH3HRH2APEX1
SCHEMBL22265138 0.70 TAAR1 (0.47) HRH4HRH1TAAR1SMN1; SMN2
Hydrochloric Acid SCHEMBL35210959 0.69 HRH1 (0.50) HRH4HRH1TAAR1HRH3HRH2
Hydrochloric Acid SCHEMBL3888095 0.69 HRH1 (0.50) HRH4HRH1TAAR1HRH3HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017029602-A2 COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-02-23 WO disclosed