SCHEMBL18544466

SCHEMBL18544466

O=C1COc2ncc(CNC3CCCCC3)nc2N1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 17/20 0.41
KCNQ1 P51787 1/20 0.41
CACNA1C Q13936 1/20 0.41
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18544246 0.76 KCNH2 (0.37) KCNH2
SCHEMBL18542847 0.75 NR3C2 (0.34) KCNH2
SCHEMBL20679486 0.75 KCNH2 (0.55) KCNH2
SCHEMBL20679441 0.74 KCNH2 (0.53) KCNH2KCNQ1CACNA1C
SCHEMBL20679263 0.74 KCNH2 (0.53) KCNH2KCNQ1CACNA1C
SCHEMBL20679510 0.74 KCNH2 (0.49) KCNH2KCNQ1CACNA1C
SCHEMBL18544254 0.74 KCNH2 (0.58) KCNH2
SCHEMBL20679241 0.74 KCNH2 (0.66) KCNH2
SCHEMBL20679511 0.74 KCNH2 (0.56) KCNH2KCNQ1CACNA1C
SCHEMBL18542787 0.74 KCNH2 (0.58) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017029602-A2 COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-02-23 WO disclosed