SCHEMBL18544475

SCHEMBL18544475

CC(C)(C)OC(=O)N[C@@H]1CC[C@@H](NC(=O)OCc2ccccc2)[C@H](O)C1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.54
GAA P10253 1/20 0.54
CPB1 P15086 2/20 0.53
TSHR P16473 1/20 0.52
KMT2A Q03164 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
KDM1A O60341 1/20 0.51
MAOB P27338 1/20 0.51
TLR4 O00206 1/20 0.47
EPHX1 P07099 1/20 0.46
DPP4 P27487 3/20 0.46
DPP7 Q9UHL4 3/20 0.46
KCNH2 Q12809 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
ACHE P22303 1/20 0.46
CCR2 P41597 1/20 0.46
CTSL P07711 2/20 0.45
SYK P43405 1/20 0.45
CTSB P07858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23871461 1.00 ALDH1A1 (0.54) ALDH1A1GAACPB1TSHRKMT2A
SCHEMBL3892622 1.00 ALDH1A1 (0.54) ALDH1A1GAACPB1TSHRKMT2A
SCHEMBL18544476 1.00 ALDH1A1 (0.54) ALDH1A1GAACPB1TSHRKMT2A
SCHEMBL18544185 1.00 ALDH1A1 (0.54) ALDH1A1GAACPB1TSHRKMT2A
SCHEMBL18544213 1.00 ALDH1A1 (0.54) ALDH1A1GAACPB1TSHRKMT2A
SCHEMBL24226875 0.91 ALDH1A1 (0.54) ALDH1A1GAACPB1TSHRKMT2A
SCHEMBL3889255 0.91 ALDH1A1 (0.54) ALDH1A1GAACPB1TSHRKMT2A
SCHEMBL23871744 0.91 ALDH1A1 (0.54) ALDH1A1GAACPB1TSHRKMT2A
SCHEMBL22241959 0.91 KMT2A (0.54) ALDH1A1GAACPB1TSHRKMT2A
SCHEMBL22241957 0.91 KMT2A (0.54) ALDH1A1GAACPB1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137616-B Antibacterial agents comprising pyrazino [2,3-b ] [1,4] oxazin-3-ones or related ring systems 葛兰素史克知识产权开发有限公司 2020-06-26 CN disclosed
WO-2017029602-A2 COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-02-23 WO disclosed