SCHEMBL1855839

SCHEMBL1855839

CCOC(=O)c1cc(F)cc(-c2ccc(F)c3cc(CBr)sc23)c1.CCOC(=O)c1cc(F)cc(-c2ccc(F)c3cc(CO)sc23)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 1/20 0.36
TRPM8 Q7Z2W7 2/20 0.35
KDM4E B2RXH2 2/20 0.35
NPC1 O15118 2/20 0.35
MAPT P10636 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
MAPK14 Q16539 2/20 0.34
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CDC7 O00311 1/20 0.33
DBF4 Q9UBU7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3200799 0.96 GPR52 (0.38) GPR52TRPM8KDM4ENPC1MAPT
SCHEMBL1851614 0.95 GPR52 (0.38) GPR52TRPM8KDM4ENPC1MAPT
SCHEMBL1851317 0.89 GPR52 (0.43) GPR52TRPM8NPC1MAPTRAB9A
SCHEMBL1859911 0.87 GPR52 (0.46) GPR52NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL1852550 0.85 GPR52 (0.46) GPR52TRPM8NPC1MAPTRAB9A
SCHEMBL1854460 0.84 NPC1 (0.36) GPR52TRPM8KDM4ENPC1MAPT
SCHEMBL1850410 0.84 GPR52 (0.47) GPR52TRPM8NPC1MAPTRAB9A
SCHEMBL1850115 0.82 GPR52 (0.44) GPR52NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL1849690 0.81 GPR52 (0.49) GPR52TRPM8KDM4ENPC1MAPT
SCHEMBL1851411 0.80 NPC1 (0.37) GPR52KDM4ENPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed