SCHEMBL18567367

SCHEMBL18567367

CNC(=O)c1ccc2[nH]c3c(c2c1)C(C)(C)Cc1c[nH]nc1-3

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 4/20 0.43
TLR8 Q9NR97 2/20 0.42
TLR7 Q9NYK1 2/20 0.42
TLR9 Q9NR96 1/20 0.40
CSNK1D P48730 1/20 0.37
CCNC P24863 4/20 0.35
CDK8 P49336 4/20 0.35
TTK P33981 1/20 0.35
CHEK1 O14757 1/20 0.34
RET P07949 2/20 0.34
PLK4 O00444 1/20 0.34
PLK1 P53350 1/20 0.34
NR1H4 Q96RI1 1/20 0.34
KDR P35968 1/20 0.33
CCNB2 O95067 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
MDH2 P40926 1/20 0.33
GSK3B P49841 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14731537 0.88 CCNB2 (0.44) MAPKAPK2CCNB2CDK1CCNB1MDH2
SCHEMBL14731397 0.88 KDM4E (0.40) MAPKAPK2NR1H4CCNB2CDK1CCNB1
SCHEMBL14731482 0.87 MAPKAPK2 (0.41) MAPKAPK2TTKNR1H4KDM4EGAA
SCHEMBL18567380 0.87 MAPKAPK2 (0.41) MAPKAPK2TLR8TLR7TLR9CSNK1D
SCHEMBL14731476 0.86 PARP1 (0.42) MAPKAPK2TLR8TLR7TLR9KDM4E
SCHEMBL14731483 0.86 RAB9A (0.39) MAPKAPK2TLR8TLR7TLR9
SCHEMBL18567602 0.85 MAPKAPK2 (0.44) MAPKAPK2TLR8TLR7TLR9CSNK1D
SCHEMBL14731478 0.85 RAB9A (0.42) TLR8TLR7TLR9
SCHEMBL14731538 0.85 RAB9A (0.45) MAPKAPK2TLR8TLR7TLR9CHEK1
SCHEMBL14731484 0.84 SMYD3 (0.49) TLR8TLR7TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2748167-B1 HEPATITIS C INHIBITOR COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2017-03-01 EP disclosed