SCHEMBL18569145

SCHEMBL18569145

CSC(C)CC(=O)N(O)c1sc(-c2cccnc2)nc1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.44
CYP3A4 P08684 3/20 0.44
CYP2C19 P33261 2/20 0.42
LMNA P02545 1/20 0.42
KDM4E B2RXH2 7/20 0.41
MAPT P10636 5/20 0.41
ALDH1A1 P00352 4/20 0.41
POLB P06746 2/20 0.41
CDC7 O00311 2/20 0.39
DBF4 Q9UBU7 2/20 0.39
GFER P55789 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
HSD17B10 Q99714 3/20 0.37
HTT P42858 1/20 0.37
TSHR P16473 1/20 0.36
FBP1 P09467 1/20 0.36
ALOX5 P09917 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13048826 0.90 CYP1A2 (0.44) CYP1A2CYP3A4CYP2C19LMNAKDM4E
SCHEMBL13048774 0.88 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C19LMNAKDM4E
SCHEMBL18569340 0.80 CYP1A2 (0.47) CYP1A2CYP3A4CYP2C19LMNAKDM4E
SCHEMBL13048022 0.80 CYP1A2 (0.44) CYP1A2CYP3A4CYP2C19LMNAKDM4E
SCHEMBL17589862 0.79 ALDH1A1 (0.41) CYP1A2CYP3A4CYP2C19LMNAKDM4E
SCHEMBL17589957 0.79 CYP1A2 (0.46) CYP1A2CYP3A4CYP2C19LMNAKDM4E
SCHEMBL13048343 0.78 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C19LMNAKDM4E
SCHEMBL13074954 0.78 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C19LMNAKDM4E
SCHEMBL13048841 0.76 KDM4E (0.43) CYP1A2CYP3A4CYP2C19LMNAKDM4E
SCHEMBL16660143 0.76 CYP1A2 (0.47) CYP1A2CYP3A4CYP2C19LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614826-B1 Process for preparation of thiazole derivatives DOW AGROSCIENCES LLC (US) 2017-03-01 EP disclosed