SCHEMBL1856929

SCHEMBL1856929

COC(=O)c1ccc(OCC2CC2)cc1Cl

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 5/20 0.50
PARP15 Q460N3 4/20 0.50
ACACB O00763 11/20 0.47
PARP2 Q9UGN5 1/20 0.46
SCN9A Q15858 2/20 0.45
ACACA Q13085 4/20 0.43
CYP2C9 P11712 3/20 0.43
CYP3A4 P08684 2/20 0.43
CNR1 P21554 1/20 0.43
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21434685 0.88 PRKAB2 (0.47) PARP10PARP15ACACB
SCHEMBL8903105 0.84 CA12 (0.55) PARP10PARP15ACACBPARP2SCN9A
SCHEMBL1854146 0.84 PARP10 (0.51) PARP10PARP15ACACBPARP2SCN9A
SCHEMBL15969380 0.84 PARP10 (0.50) PARP10PARP15ACACBPARP2
SCHEMBL3225627 0.83 PARP10 (0.67) PARP10PARP15ACACBPARP2SCN9A
SCHEMBL1856415 0.83 PARP10 (0.64) PARP10PARP15ACACBPARP2SCN9A
SCHEMBL26126220 0.83 PARP10 (0.53) PARP10PARP15ACACBPARP2SCN9A
SCHEMBL6301208 0.81 PARP10 (0.56) PARP10PARP15PARP2
SCHEMBL21447016 0.81 TDP1 (0.51)
SCHEMBL2089720 0.80 PARP10 (0.50) PARP10PARP15ACACBPARP2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323988-A1 ALPHA7 NICOTINIC ACETYLCHOLINE RECEPTOR INHIBITORS Wyeth LLC (US) 2011-05-25 EP disclosed
WO-2010009290-A1 ALPHA7 NICOTINIC ACETYLCHOLINE RECEPTOR INHIBITORS WYETH (US) 2010-01-21 WO disclosed
WO-2009091832-A1 SYNTHESIS OF PYRAZOLES WYETH (US) 2009-07-23 WO disclosed