SCHEMBL18570980

SCHEMBL18570980

C=Cc1ccc(C(F)(F)F)cc1CCC(C)C

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 4/20 0.39
SLC6A4 P31645 4/20 0.39
PDE2A O00408 3/20 0.36
SLC6A3 Q01959 2/20 0.36
SCN10A Q9Y5Y9 1/20 0.35
S1PR1 P21453 2/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
IDO1 P14902 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HRH4 Q9H3N8 1/20 0.32
KCNH2 Q12809 2/20 0.32
TMEM97 Q5BJF2 2/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
BACE1 P56817 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24061603 0.79 PDE2A (0.39) SLC6A4PDE2AS1PR1HTR2AIDO1
SCHEMBL14131082 0.76 FFAR4 (0.43) SLC6A2SLC6A4PDE2AKCNH2TMEM97
SCHEMBL3678271 0.76 IDO1 (0.37) PDE2AIDO1ALDH1A1CYP3A4CYP2D6
SCHEMBL30233883 0.75 CYP1A1 (0.43) PDE2ASCN10ABACE1KDM4E
SCHEMBL25026056 0.75 CYP1A1 (0.43) PDE2ASCN10ABACE1KDM4E
SCHEMBL28173592 0.74 SLC6A4 (0.51) SLC6A2SLC6A4PDE2ASLC6A3HTR2A
SCHEMBL18570695 0.74 CSNK1D (0.38) SLC6A2SLC6A4PDE2AIDO1CYP2D6
SCHEMBL20344484 0.72 RXFP1 (0.36) SLC6A2SLC6A4ALDH1A1KCNH2TMEM97
SCHEMBL4263679 0.72 SLC6A2 (0.38) SLC6A2SLC6A4SLC6A3HTR2BALDH1A1
SCHEMBL15067318 0.71 ACP1 (0.38) IDO1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2953931-B1 PYRIDONE AMIDES AS MODULATORS OF SODIUM CHANNELS VERTEX PHARMA (US) 2017-03-01 EP disclosed