SCHEMBL18587397

SCHEMBL18587397

Cc1ccc(N2CCc3cc(OCc4ccccc4)ccc3[C@@H](O)[C@H]2C)cc1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 2/20 0.52
MMP2 P08253 2/20 0.52
MMP7 P09237 2/20 0.52
MMP9 P14780 2/20 0.52
MMP12 P39900 2/20 0.52
MMP14 P50281 2/20 0.52
MMP15 P51511 2/20 0.52
MMP16 P51512 2/20 0.52
MMP26 Q9NRE1 2/20 0.52
GRIN1 Q05586 10/20 0.50
GRIN2B Q13224 10/20 0.50
HRH3 Q9Y5N1 4/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18587613 1.00 MMP1 (0.52) MMP1MMP2MMP7MMP9MMP12
SCHEMBL3394741 0.82 MMP1 (0.70) MMP1MMP2MMP7MMP9MMP12
SCHEMBL3392159 0.82 MMP1 (0.70) MMP1MMP2MMP7MMP9MMP12
SCHEMBL3397104 0.82 MMP1 (0.70) MMP1MMP2MMP7MMP9MMP12
SCHEMBL3393324 0.82 MMP1 (0.70) MMP1MMP2MMP7MMP9MMP12
SCHEMBL3807794 0.80 HRH3 (0.58) MMP1MMP2MMP7MMP9MMP12
SCHEMBL3422815 0.78 MAOB (0.54) MMP1MMP2MMP7MMP9MMP12
SCHEMBL3422819 0.78 MAOB (0.54) MMP1MMP2MMP7MMP9MMP12
SCHEMBL3397537 0.77 GRIN1 (0.66) GRIN1GRIN2BHRH3
SCHEMBL13069934 0.77 GRIN1 (0.66) GRIN1GRIN2BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3344257-A1 NR2B SELECTIVE NMDA-RECEPTOR ANTAGONISTS FOR TREATMENT OF IMMUNE-MEDIATED INFLAMMATORY DISEASES Westfälische Wilhelms-Universität Münster (DE) 2018-07-11 EP disclosed
WO-2017036880-A1 NR2B SELECTIVE NMDA-RECEPTOR ANTAGONISTS FOR TREATMENT OF IMMUNE-MEDIATED INFLAMMATORY DISEASES Westfälische Wilhelms-Universität Münster (DE) 2017-03-09 WO disclosed