SCHEMBL18593151

SCHEMBL18593151

COC1CCN(c2cc[nH]n2)CC1(C)O

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.40
TYK2 P29597 3/20 0.40
LRRK2 Q5S007 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18593193 0.86 JAK2 (0.38) JAK2TYK2
SCHEMBL18592922 0.83 JAK2 (0.37) JAK2TYK2LRRK2
SCHEMBL18593175 0.82 JAK2 (0.38) JAK2TYK2LRRK2
SCHEMBL18592869 0.74 KHK (0.41) JAK2TYK2LRRK2
SCHEMBL18592873 0.74 KHK (0.41) JAK2TYK2LRRK2
SCHEMBL18592872 0.74 KHK (0.41) JAK2TYK2LRRK2
SCHEMBL23008368 0.73 MAP4K4 (0.45) LRRK2
SCHEMBL18593206 0.72 JAK2 (0.37) JAK2TYK2
SCHEMBL20380485 0.71 LRRK2 (0.39) JAK2TYK2LRRK2
SCHEMBL18592814 0.71 LRRK2 (0.39) JAK2TYK2LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4327809-A2 TYK2 INHIBITORS AND USES THEREOF Takeda Pharmaceutical Company Limited (JP) 2024-02-28 EP disclosed
EP-3344624-B1 TYK2 INHIBITORS AND USES THEREOF NIMBUS LAKSHMI INC (US) 2023-10-25 EP disclosed
US-20210047319-A1 TYK2 INHIBITORS AND USES THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-02-18 US disclosed
US-10781204-B2 TYK2 inhibitors and uses thereof NIMBUS LAKSHMI, INC. (US) 2020-09-22 US disclosed
US-10023571-B2 TYK2 inhibitors and uses thereof Nimbus Lakshimi, Inc. (US) 2018-07-17 US disclosed
US-10023571-B2 TYK2 inhibitors and uses thereof Nimbus Lakshimi, Inc. (US) 2018-07-17 US disclosed
US-20170066763-A1 TYK2 INHIBITORS AND USES THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-03-09 US disclosed
US-20170066763-A1 TYK2 INHIBITORS AND USES THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-03-09 US disclosed
WO-2017040757-A1 TYK2 INHIBITORS AND USES THEREOF NIMBUS LAKSHMI, INC. (US) 2017-03-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170066763-A1 TYK2 INHIBITORS AND USES THEREOF TYK2, JAK2, JAK1 JAK2 2/4885TYK2 1/4885LRRK2 269/4885
US-10023571-B2 TYK2 inhibitors and uses thereof TYK2, JAK1, JAK2 JAK2 3/4885TYK2 1/4885LRRK2 259/4885
US-20210047319-A1 TYK2 INHIBITORS AND USES THEREOF TYK2, JAK2, JAK1 JAK2 2/4885TYK2 1/4885LRRK2 269/4885
US-10781204-B2 TYK2 inhibitors and uses thereof TYK2, JAK1, JAK2 JAK2 3/4885TYK2 1/4885LRRK2 259/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.