SCHEMBL18595010

SCHEMBL18595010

CCNC(=O)c1csc(NC(=O)NCc2ccccc2)n1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 13/20 0.59
ROCK1 Q13464 13/20 0.59
SMN1; SMN2 Q16637 2/20 0.49
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
HIF1A Q16665 1/20 0.48
GAA P10253 1/20 0.47
MMP3 P08254 1/20 0.47
LCK P06239 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7141146 0.88 ROCK2 (0.59) ROCK2ROCK1SMN1; SMN2HIF1AMMP3
SCHEMBL18595025 0.86 ROCK2 (0.55) ROCK2ROCK1SMN1; SMN2HIF1AMMP3
SCHEMBL6880276 0.86 ROCK2 (0.65) ROCK2ROCK1MMP3
SCHEMBL15145661 0.86 PPID (0.60) ROCK2ROCK1SMN1; SMN2NPC1RAB9A
SCHEMBL6316630 0.84 ROCK2 (0.62) ROCK2ROCK1MMP3
SCHEMBL7140708 0.83 ROCK2 (0.52) ROCK2ROCK1SMN1; SMN2NPC1RAB9A
SCHEMBL7301734 0.83 SMN1; SMN2 (0.67) ROCK2ROCK1SMN1; SMN2NPC1RAB9A
SCHEMBL7140468 0.83 ROCK2 (0.54) ROCK2ROCK1HIF1AGAA
SCHEMBL27575975 0.83 ROCK2 (0.54) ROCK2ROCK1SMN1; SMN2MMP3LCK
SCHEMBL27558247 0.83 ROCK2 (0.54) ROCK2ROCK1SMN1; SMN2MMP3LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9586916-B2 Integrin antagonist conjugates for targeted delivery to cells expressing alpha-V-beta-3 HOFFMANN-LA ROCHE INC. (US) 2017-03-07 US disclosed