SCHEMBL1860029

SCHEMBL1860029

CN(CCO)C(=O)c1ccc(C(F)(F)F)c(-c2ccc3c(Nc4ncc(C(F)(F)F)cn4)ccnc3n2)n1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 17/20 0.59
MAPK3 P27361 1/20 0.47
SCN9A Q15858 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12666844 0.91 TRPV1 (0.51) TRPV1MAPK3SCN9A
SCHEMBL1862801 0.89 TRPV1 (0.47) TRPV1MAPK3SCN9A
SCHEMBL1858241 0.86 TRPV1 (0.58) TRPV1MAPK3
SCHEMBL1864049 0.85 TRPV1 (0.46) TRPV1SCN9A
SCHEMBL1856817 0.84 TRPV1 (0.69) TRPV1MAPK3
SCHEMBL1858558 0.84 TRPV1 (0.66) TRPV1MAPK3SCN9A
SCHEMBL12664963 0.82 TRPV1 (0.50) TRPV1MAPK3
SCHEMBL1866310 0.80 TRPV1 (0.66) TRPV1MAPK3
SCHEMBL12666701 0.79 TRPV1 (0.42) TRPV1SCN9A
SCHEMBL1863478 0.79 TRPV1 (0.74) TRPV1MAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7935702-B2 Substituted biaryl quinolin-4-ylamine analogues NEUROGEN CORPORATION (US) 2011-05-03 US disclosed
US-7935702-B2 Substituted biaryl quinolin-4-ylamine analogues NEUROGEN CORPORATION (US) 2011-05-03 US disclosed