SCHEMBL18601432

SCHEMBL18601432

O=C(C=Cc1ccccn1)c1cc(OCCc2ccc(F)cc2)ccc1O

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.56
MAPT P10636 3/20 0.56
HSP90AA1 P07900 2/20 0.56
ALDH1A1 P00352 2/20 0.56
NPSR1 Q6W5P4 1/20 0.56
PPARA Q07869 1/20 0.46
MAOB P27338 3/20 0.46
AR P10275 2/20 0.45
SIRT2 Q8IXJ6 1/20 0.44
CYSLTR2 Q9NS75 1/20 0.42
CYSLTR1 Q9Y271 1/20 0.42
CYP1B1 Q16678 1/20 0.42
MAOA P21397 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18601431 1.00 KDM4E (0.56) KDM4EMAPTHSP90AA1ALDH1A1NPSR1
SCHEMBL2840220 0.93 KDM4E (0.59) KDM4EMAPTHSP90AA1ALDH1A1NPSR1
SCHEMBL2840222 0.93 KDM4E (0.59) KDM4EMAPTHSP90AA1ALDH1A1NPSR1
SCHEMBL751930 0.91 KDM4E (0.57) KDM4EMAPTHSP90AA1ALDH1A1NPSR1
SCHEMBL751929 0.91 KDM4E (0.57) KDM4EMAPTHSP90AA1ALDH1A1NPSR1
SCHEMBL17907496 0.89 CYSLTR2 (0.56) KDM4EMAPTHSP90AA1ALDH1A1NPSR1
SCHEMBL17907495 0.89 CYSLTR2 (0.56) KDM4EMAPTHSP90AA1ALDH1A1NPSR1
SCHEMBL752857 0.81 CYSLTR2 (0.62) KDM4EMAPTHSP90AA1ALDH1A1NPSR1
SCHEMBL752858 0.81 CYSLTR2 (0.62) KDM4EMAPTHSP90AA1ALDH1A1NPSR1
SCHEMBL2790877 0.80 KDM4E (0.65) KDM4EMAPTHSP90AA1ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2266958-B1 Antiviral agent SHIONOGI & CO (JP) 2017-03-15 EP disclosed