SCHEMBL18601899

SCHEMBL18601899

COC1=CCC(N2CN(Cc3cccc(C(=O)O)c3)C(=O)C23CCN(CCCn2c(=O)sc4ccccc42)CC3)C=C1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.41
HTR7 P34969 5/20 0.41
MEN1 O00255 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HRH2 P25021 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18602007 0.88 P2RX7 (0.41) HTR1AHTR7MEN1TP53CYP1A2
SCHEMBL318607 0.81 MEN1 (0.49) HTR1AHTR7MEN1TP53CYP1A2
SCHEMBL318993 0.80 MEN1 (0.56) HTR1AHTR7MEN1TP53CYP1A2
SCHEMBL18601842 0.79 CYP1A2 (0.43) HTR7MEN1TP53CYP1A2CYP3A4
SCHEMBL318732 0.78 MEN1 (0.53) HTR1AHTR7MEN1TP53CYP1A2
SCHEMBL10248483 0.76 MEN1 (0.54) HTR1AHTR7MEN1TP53CYP1A2
SCHEMBL319183 0.76 MEN1 (0.47) HTR1AHTR7MEN1TP53CYP1A2
SCHEMBL18601799 0.75 P2RX7 (0.44) HTR7MEN1TP53CYP1A2CYP3A4
SCHEMBL318646 0.70 KCNH2 (0.51) HTR1AHTR7MEN1TP53CYP1A2
SCHEMBL318643 0.69 MEN1 (0.57) MEN1TP53CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3138841-A1 D2 ANTAGONISTS, METHODS OF SYNTHESIS AND METHODS OF USE Altos Therapeutics, LLC (US) 2017-03-08 EP disclosed