SCHEMBL18614740

SCHEMBL18614740

CCOC(=O)CCCN(c1cnc(-c2ccccc2)c(-c2ccccc2)n1)C(C)C

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.66
NR1I2 O75469 2/20 0.66
TBXA2R P21731 2/20 0.66
AGTR1 P30556 2/20 0.66
PTGIR P43119 2/20 0.66
PDE4D Q08499 2/20 0.66
PTGDR Q13258 2/20 0.66
DRD1 P21728 1/20 0.66
CKS1B P61024 4/20 0.59
SKP1 P63208 4/20 0.59
SKP2 Q13309 4/20 0.59
ABCB11 O95342 1/20 0.59
HTR1A P08908 1/20 0.59
CNR1 P21554 1/20 0.59
HTR2A P28223 1/20 0.59
ADRA1A P35348 1/20 0.59
OPRD1 P41143 1/20 0.59
OPRK1 P41145 1/20 0.59
HTR2B P41595 1/20 0.59
SCN5A Q14524 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21014626 0.88 ADORA3 (0.80) ADORA3NR1I2TBXA2RAGTR1PTGIR
SCHEMBL18614888 0.87 PTGIR (0.74) ADORA3NR1I2TBXA2RAGTR1PTGIR
SCHEMBL5218595 0.83 CKS1B (0.54) ADORA3NR1I2TBXA2RAGTR1PTGIR
SCHEMBL5213530 0.83 CKS1B (0.54) ADORA3NR1I2TBXA2RAGTR1PTGIR
SCHEMBL29068587 0.83 NR1I2 (0.75) ADORA3NR1I2TBXA2RAGTR1PTGIR
SCHEMBL18630465 0.82 NR1I2 (0.66) ADORA3NR1I2TBXA2RAGTR1PTGIR
SCHEMBL28690981 0.82 NR1I2 (0.66) ADORA3NR1I2TBXA2RAGTR1PTGIR
SCHEMBL18584837 0.81 NR1I2 (0.66) ADORA3NR1I2TBXA2RAGTR1PTGIR
SCHEMBL19820820 0.81 NR1I2 (0.68) ADORA3NR1I2TBXA2RAGTR1PTGIR
Acetic Acid SCHEMBL29068588 0.80 NR1I2 (0.71) ADORA3NR1I2TBXA2RAGTR1PTGIR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017042828-A2 PROCESS FOR THE PREPARATION OF SELEXIPAG AND INTERMEDIATES THEREOF MEGAFINE PHARMA (P) LTD. (IN) 2017-03-16 WO disclosed
WO-2017042828-A2 PROCESS FOR THE PREPARATION OF SELEXIPAG AND INTERMEDIATES THEREOF MEGAFINE PHARMA (P) LTD. (IN) 2017-03-16 WO disclosed