SCHEMBL18616636

SCHEMBL18616636

NC(=O)c1cc(-c2cnc3ccccc3c2)cnc1N

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.60
PIK3CB P42338 1/20 0.55
PARP1 P09874 2/20 0.52
MAP4K4 O95819 2/20 0.51
MKNK2 Q9HBH9 2/20 0.51
CSNK1G2 P78368 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
MAP4K5 Q9Y4K4 1/20 0.51
PDGFRB P09619 2/20 0.50
PDGFRA P16234 2/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
CYP2A6 P11509 1/20 0.48
BIRC5 O15392 1/20 0.47
MGAM O43451 1/20 0.46
HSP90AA1 P07900 3/20 0.46
MTOR P42345 1/20 0.46
PIK3CD O00329 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18615848 0.83 MKNK1 (0.61) IKBKBPIK3CBPARP1MAP4K4MKNK2
SCHEMBL17610489 0.82 IKBKB (0.56) IKBKBPARP1MAP4K4MKNK2CSNK1G2
SCHEMBL14917448 0.82 IKBKB (0.56) IKBKBPARP1MAP4K4MKNK2CSNK1G2
SCHEMBL18615835 0.81 CHEK2 (0.64) IKBKBPIK3CBPARP1MAP4K4MKNK2
SCHEMBL995473 0.81 PARP1 (0.54) IKBKBPARP1MAP4K4MKNK2CSNK1G2
SCHEMBL31127659 0.81 PARP1 (0.54) IKBKBPARP1MAP4K4MKNK2CSNK1G2
SCHEMBL17610492 0.79 IKBKB (0.49) IKBKBPARP1MAP4K4MKNK2CSNK1G2
SCHEMBL26613435 0.79 CA12 (0.60) PARP1MAP4K4MKNK2CSNK1G2CLK4
SCHEMBL4686366 0.79 IKBKB (0.67) IKBKBPARP1MAP4K4MKNK2CSNK1G2
SCHEMBL31032045 0.77 PARP1 (0.50) IKBKBPARP1MAP4K4MKNK2CSNK1G2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3344613-B1 HETEROARYL COMPOUNDS AND THEIR USE AS THERAPEUTIC DRUGS DONG A SOCIO HOLDINGS CO LTD (KR) 2020-03-04 EP disclosed
WO-2017039331-A1 HETEROARYL COMPOUNDS AND THEIR USE AS THERAPEUTIC DRUGS DONG-A SOCIO HOLDINGS CO., LTD. (KR) 2017-03-09 WO disclosed