SCHEMBL26613435

SCHEMBL26613435

NC(=O)c1ccc(-c2cnc3ccccc3c2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.60
CA1 P00915 1/20 0.60
CA2 P00918 1/20 0.60
CA9 Q16790 1/20 0.60
MKNK1 Q9BUB5 4/20 0.58
MKNK2 Q9HBH9 4/20 0.58
CHEK2 O96017 4/20 0.57
MAP4K4 O95819 2/20 0.57
RIPK1 Q13546 1/20 0.57
CSNK1G2 P78368 1/20 0.57
CLK4 Q9HAZ1 1/20 0.57
MAP4K5 Q9Y4K4 1/20 0.57
PDGFRB P09619 1/20 0.57
PDGFRA P16234 1/20 0.57
FASN P49327 1/20 0.54
TNIK Q9UKE5 1/20 0.53
MGAM O43451 1/20 0.53
PIK3CD O00329 1/20 0.51
PIK3CA P42336 1/20 0.51
PARP1 P09874 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31187396 0.88 MKNK2 (0.56) CA12CA1CA2CA9MKNK1
SCHEMBL8109340 0.86 MGAM (0.68) CA12CA1CA2CA9MKNK2
SCHEMBL30108206 0.85 MKNK2 (0.58) CA12CA1CA2CA9MKNK1
SCHEMBL944068 0.85 CSNK1G2 (0.74) CA12CA1CA2CA9MKNK2
SCHEMBL27873382 0.84 MMP1 (0.56) CA12CA1CA2CA9MKNK2
SCHEMBL29362497 0.82 MGAM (0.71) MKNK2CHEK2MAP4K4CSNK1G2CLK4
SCHEMBL23372 0.82 MGAM (0.71) MKNK2CHEK2MAP4K4CSNK1G2CLK4
Hydrochloric Acid SCHEMBL5311903 0.80 MGAM (0.69) MKNK2CHEK2MAP4K4CSNK1G2CLK4
Fluoride SCHEMBL28234122 0.80 MGAM (0.69) MKNK2CHEK2MAP4K4CSNK1G2CLK4
Hydrochloric Acid SCHEMBL28841803 0.80 MGAM (0.69) MKNK2CHEK2MAP4K4CSNK1G2CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260083723-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR AMYOTROPHIC LATERAL SCLEROSIS TORAY INDUSTRIES, INC. (JP) 2026-03-26 US disclosed
US-12570639-B2 Tetrahydroquinoline derivative and medicinal use thereof TORAY INDUSTRIES, INC. (JP) 2026-03-10 US disclosed
EP-4545079-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR AMYOTROPHIC LATERAL SCLEROSIS Toray Industries, Inc. (JP) 2025-04-30 EP disclosed
CN-119403554-A Therapeutic or prophylactic agent for amyotrophic lateral sclerosis 东丽株式会社 2025-02-07 CN disclosed
US-20240116903-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF TORAY INDUSTRIES, INC. (JP) 2024-04-11 US disclosed
WO-2023249107-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR PERIPHERAL NERVE DISORDER 東レ株式会社 2023-12-28 WO disclosed
WO-2023249106-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR AMYOTROPHIC LATERAL SCLEROSIS 東レ株式会社 2023-12-28 WO disclosed
WO-2023249105-A1 THERAPEUTIC AGENT OR PREVENTIVE AGENT FOR DRUG-INDUCED MYOCARDIAL DISORDERS 東レ株式会社 2023-12-28 WO disclosed
EP-4269392-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF Toray Industries, Inc. (JP) 2023-11-01 EP disclosed
EP-4269392-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF Toray Industries, Inc. (JP) 2023-11-01 EP disclosed
CN-116648245-A Tetrahydroquinoline derivative and medical application thereof 东丽株式会社 2023-08-25 CN disclosed
WO-2022138888-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF 東レ株式会社 2022-06-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240116903-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF AIFM2, TXNRD2, NFE2L2 CA12 4293/4885CA1 3259/4885CA2 2071/4885
US-20260083723-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR AMYOTROPHIC LATERAL SCLEROSIS AIFM2, GPX1, SOD1 CA12 3763/4885CA1 1020/4885CA2 1110/4885
US-12570639-B2 Tetrahydroquinoline derivative and medicinal use thereof AIFM2, GPX1, GPX4 CA12 3197/4885CA1 1600/4885CA2 1497/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.