SCHEMBL18618596

SCHEMBL18618596

Cc1cc(OCc2nn(C(=O)OC(C)(C)C)c3nc(F)ccc23)c(C(C)(C)C)cc1Cl

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
F2RL1 P55085 1/20 0.32
PTGES O14684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29588571 1.00 F2RL1 (0.32) F2RL1PTGES
SCHEMBL29588959 0.92 F2RL1 (0.33) F2RL1PTGES
SCHEMBL18617540 0.92 F2RL1 (0.33) F2RL1PTGES
SCHEMBL22579145 0.90 PPARG (0.32) PTGES
SCHEMBL18617547 0.86 POLB (0.34) PTGES
SCHEMBL29587617 0.86 POLB (0.34) PTGES
SCHEMBL22579143 0.82 PTGES (0.32) PTGES
SCHEMBL18617507 0.78
SCHEMBL18617537 0.75 SYK (0.40)
SCHEMBL29588508 0.75 SYK (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11352330-B2 Phenoxymethyl derivatives HOFFMANN-LA ROCHE INC. (US) 2022-06-07 US disclosed
US-20200339522-A1 PHENOXYMETHYL DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2020-10-29 US disclosed
EP-3344619-B1 PHENOXYMETHYL DERIVATIVES HOFFMANN LA ROCHE (CH) 2020-10-28 EP disclosed
US-10640472-B2 Phenoxymethyl derivatives HOFFMAN-LA ROCHE INC. (US) 2020-05-05 US disclosed
US-20180201588-A1 PHENOXYMETHYL DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2018-07-19 US disclosed
US-20180201588-A1 PHENOXYMETHYL DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2018-07-19 US disclosed
WO-2017037146-A1 PHENOXYMETHYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2017-03-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200339522-A1 PHENOXYMETHYL DERIVATIVES CNKSR1, RB1, RCOR1 F2RL1 1990/4885PTGES 833/4885
US-10640472-B2 Phenoxymethyl derivatives CNKSR1, RB1, RCOR1 F2RL1 1990/4885PTGES 833/4885
US-20180201588-A1 PHENOXYMETHYL DERIVATIVES CNKSR1, RB1, RCOR1 F2RL1 1990/4885PTGES 833/4885
US-11352330-B2 Phenoxymethyl derivatives CNKSR1, RB1, RCOR1 F2RL1 1990/4885PTGES 833/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.