SCHEMBL18628367

SCHEMBL18628367

O=C(Nc1ccccc1-c1ccccc1)N1CCN2C(=O)N(C3CC3c3ccc(F)cc3)C(=O)C2C1

nearest known ligand 0.88

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SMO Q99835 18/20 0.88
PAX8 Q06710 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18628368 1.00 SMO (0.88) SMOPAX8KMT2ANPSR1
SCHEMBL2160744 0.94 SMO (1.00) SMO
SCHEMBL2160741 0.94 SMO (1.00) SMO
SCHEMBL2160629 0.94 SMO (1.00) SMO
SCHEMBL18628460 0.92 SMO (0.82) SMOPAX8
SCHEMBL2160672 0.91 SMO (0.88) SMO
SCHEMBL2160674 0.91 SMO (0.88) SMO
SCHEMBL18628419 0.90 SMO (0.77) SMOPAX8NPSR1
SCHEMBL18628444 0.89 SMO (0.84) SMOPAX8KMT2ANPSR1
SCHEMBL18628439 0.89 SMO (0.84) SMOPAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334683-B1 SATURATED BICYCLIC HETEROCYCLIC DERIVATIVES AS SMO ANTAGONISTS MSD ITALIA SRL (IT) 2017-03-22 EP disclosed