SCHEMBL18628419

SCHEMBL18628419

O=C(Nc1ccccc1-c1ccccc1)N1CCN2C(=O)N(C3CC3c3ccc(F)cc3F)C(=O)[C@@H]2C1

nearest known ligand 0.77

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMO Q99835 16/20 0.77
PAX8 Q06710 2/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18628367 0.90 SMO (0.88) SMOPAX8NPSR1
SCHEMBL18628368 0.90 SMO (0.88) SMOPAX8NPSR1
SCHEMBL2160744 0.87 SMO (1.00) SMO
SCHEMBL2160629 0.87 SMO (1.00) SMO
SCHEMBL2160741 0.87 SMO (1.00) SMO
SCHEMBL18628460 0.87 SMO (0.82) SMOPAX8
SCHEMBL18628497 0.85 SMO (0.77) SMOPAX8MAPK1
SCHEMBL2160672 0.83 SMO (0.88) SMO
SCHEMBL2160674 0.83 SMO (0.88) SMO
SCHEMBL18628438 0.82 SMO (0.80) SMONPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334683-B1 SATURATED BICYCLIC HETEROCYCLIC DERIVATIVES AS SMO ANTAGONISTS MSD ITALIA SRL (IT) 2017-03-22 EP disclosed