SCHEMBL18630355

SCHEMBL18630355

CN1C=Cc2ccncc2C1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.35
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32
NAMPT P43490 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28242885 0.85 SIGMAR1 (0.35) SIGMAR1PDE3BPDE3ACHRNB2CHRNA4
SCHEMBL28319871 0.74 SIGMAR1 (0.32) SIGMAR1PDE3BPDE3ACHRNB2CHRNA4
SCHEMBL28319875 0.74 PDE3B (0.34) SIGMAR1PDE3BPDE3ACHRNB2CHRNA4
SCHEMBL3818780 0.73 NAMPT (0.35) PDE3BPDE3ANAMPT
SCHEMBL30385312 0.72 HDAC3 (0.41)
SCHEMBL1564351 0.72 HDAC3 (0.41)
SCHEMBL31691807 0.71 HDAC2 (0.36) PDE3BPDE3ANAMPT
SCHEMBL28319864 0.71 CA12 (0.35) SIGMAR1PDE3BPDE3ANAMPT
Iodide SCHEMBL4322466 0.71 HDAC3 (0.40)
Iodide SCHEMBL11870312 0.71 HDAC3 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2997021-B1 NEW SOMATOSTATIN RECEPTOR SUBTYPE 4 (SSTR4) AGONISTS CENTREXION THERAPEUTICS CORP (US) 2017-12-20 EP disclosed
EP-3141542-A1 SUBSTITUTED BENZALDEHYDE COMPOUNDS AND METHODS FOR THEIR USE IN INCREASING TISSUE OXYGENATION Global Blood Therapeutics, Inc. (US) 2017-03-15 EP disclosed