SCHEMBL18635601

SCHEMBL18635601

CCC(O)C(C)(O)c1ccccn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
CHRM3 P20309 1/20 0.38
BLM P54132 2/20 0.37
CYP2D6 P10635 1/20 0.37
AHR P35869 1/20 0.37
CHRM2 P08172 1/20 0.37
KCNA5 P22460 1/20 0.36
HDAC6 Q9UBN7 2/20 0.36
CYP1A2 P05177 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TSHR P16473 2/20 0.35
SLC22A2 O15244 1/20 0.35
SLC22A1 O15245 1/20 0.35
PGR P06401 1/20 0.35
THRB P10828 1/20 0.35
ADRB3 P13945 1/20 0.35
OPRK1 P41145 1/20 0.35
PMP22 Q01453 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17490338 1.00 SMN1; SMN2 (0.50) SMN1; SMN2L3MBTL1CHRM3BLMCYP2D6
SCHEMBL17490349 0.84 SMN1; SMN2 (0.52) SMN1; SMN2L3MBTL1CHRM3BLMCYP2D6
SCHEMBL16132385 0.83 SMN1; SMN2 (0.47) SMN1; SMN2L3MBTL1CHRM3BLMCYP2D6
SCHEMBL17490360 0.83 SMN1; SMN2 (0.50) SMN1; SMN2L3MBTL1CHRM3BLMCYP2D6
SCHEMBL16132477 0.81 SMN1; SMN2 (0.44) SMN1; SMN2L3MBTL1CHRM3BLMCYP2D6
SCHEMBL16132483 0.81 SMN1; SMN2 (0.44) SMN1; SMN2L3MBTL1CHRM3BLMCYP2D6
SCHEMBL16132485 0.80 SMN1; SMN2 (0.47) SMN1; SMN2L3MBTL1CHRM3BLMAHR
SCHEMBL16132387 0.80 SMN1; SMN2 (0.43) SMN1; SMN2L3MBTL1CHRM3BLMCYP2D6
SCHEMBL16132352 0.80 SMN1; SMN2 (0.43) SMN1; SMN2L3MBTL1CHRM3BLMCYP2D6
SCHEMBL12238622 0.78 SMN1; SMN2 (0.57) SMN1; SMN2L3MBTL1CHRM3BLMCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2978759-B1 BENZIMIDAZOLONE DERIVATIVES AS BROMODOMAIN INHIBITORS GILEAD SCIENCES INC (US) 2017-03-15 EP disclosed