SCHEMBL18635641

SCHEMBL18635641

NC(O)(c1ccccn1)C1CCCCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
MEN1 O00255 5/20 0.41
KMT2A Q03164 4/20 0.41
CHRM3 P20309 3/20 0.40
CHRM2 P08172 2/20 0.40
HPGD P15428 2/20 0.39
CYP1A2 P05177 2/20 0.38
GRM5 P41594 1/20 0.38
RECQL P46063 1/20 0.38
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37
GAA P10253 1/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TP53 P04637 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18635455 0.98 SMN1; SMN2 (0.50) SMN1; SMN2L3MBTL1MEN1KMT2ACHRM3
SCHEMBL8018028 0.83 SMN1; SMN2 (0.42) SMN1; SMN2L3MBTL1MEN1KMT2ACHRM3
SCHEMBL16132528 0.80 SMN1; SMN2 (0.48) SMN1; SMN2L3MBTL1MEN1KMT2ACHRM3
SCHEMBL3122492 0.80 SMN1; SMN2 (0.40) SMN1; SMN2L3MBTL1MEN1KMT2ACHRM3
SCHEMBL16132392 0.80 SMN1; SMN2 (0.44) SMN1; SMN2L3MBTL1MEN1KMT2ACHRM3
SCHEMBL17490363 0.78 L3MBTL1 (0.50) SMN1; SMN2L3MBTL1MEN1KMT2ACHRM3
SCHEMBL21742369 0.78 NR1I2 (0.46) SMN1; SMN2L3MBTL1MEN1KMT2ACHRM3
SCHEMBL16132505 0.78 SMN1; SMN2 (0.46) SMN1; SMN2L3MBTL1MEN1KMT2ACHRM3
SCHEMBL16291257 0.76 MEN1 (0.50) SMN1; SMN2L3MBTL1MEN1KMT2ACHRM3
Hydrochloric Acid SCHEMBL11680499 0.76 NPY2R (0.46) SMN1; SMN2L3MBTL1MEN1KMT2ACHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2978759-B1 BENZIMIDAZOLONE DERIVATIVES AS BROMODOMAIN INHIBITORS GILEAD SCIENCES INC (US) 2017-03-15 EP disclosed